Aza-THIP is a selective and moderately potent GABAA-ρ (GABAC receptor) antagonist related to gaboxadol (THIP). Unlike gaboxadol, it is virtually inactive at the GABAA receptor. The drug was first described in the scientific literature by Povl Krogsgaard-Larsen and colleagues by 1979.
See also Thio-THIP Iso-THIP THAZ
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