An adenosine reuptake inhibitor (AdoRI) is a type of drug which acts as a reuptake inhibitor for the purine nucleoside and neurotransmitter adenosine by blocking the action of one or more of the equilibrative nucleoside transporters (ENTs). This in turn leads to increased extracellular concentrations of adenosine and therefore an increase in adenosinergic neurotransmission.

List of AdoRIs

Benzodiazepines Calcium channel blockers Carisoprodol Cilostazol Cyclobenzaprine Dilazep Dipyridamole Estradiol Ethanol Hexobendine Hydroxyzine Inosine KF24345 Meprobamate Nitrobenzylthioguanosine Nitrobenzylthioinosine Papaverine Pentoxifylline Phenothiazines Phenytoin Progesterone Propentofylline Puromycin R75231 RE 102 BS Soluflazine Toyocamycin Tracazolate Tricyclic antidepressants

See also Adenosinergic Reuptake inhibitor

References